Chemistry

Enzymes build carbon-sulfur bonds using a split carbene transfer pathway

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This research demonstrates that engineered enzymes can catalyze stereoselective carbon-sulfur bond formation through a carbene transfer mechanism. The study reveals that the enzyme operates through a dichotomic pathway, meaning it can proceed through two distinct mechanistic routes to form C(sp3)-S bonds with high stereoselectivity. This represents a novel enzymatic approach to creating chiral organosulfur compounds, which are important building blocks in pharmaceutical chemistry.


This enzymatic method offers a more sustainable and selective alternative to traditional metal-based catalysts for synthesizing sulfur-containing molecules. The ability to control stereochemistry through enzyme engineering has significant implications for pharmaceutical development, where the three-dimensional arrangement of atoms critically affects drug efficacy and safety.


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Journal of the American Chemical Society
DOI: 10.1021/jacs.6c02960

Source: [ASAP] Enzyme-Catalyzed Stereoselective C(sp3)–S Bond Formation via a Dichotomic Carbene Transfer Mechanism